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European Patent (TR Translation)

Platelet Agregasyonunun Tedavi Edilmesine Yönelik Proteaz İle Aktive Edilen Reseptör 4 (Par4) İnhibitörleri Olarak İmidazotiyadiazol Ve İmidazopirazin Deriveleri.

Invention Abstract

Mevcut buluş, W, Y, R0, R2, R4, R5, R6, R7, X1, X2, X3 ve X4'ün burada tanımlanan gibi olduğu Formülün (I) tiyozol bileşiklerini veya bir stereoizomeri, totomeri, farmasötik olarak kabul edilebilir bir tuzu, ön ilaç ester veya solvat formunu sağlar, burada değişkenlerin tümü burada tanımlanan gibidir. Bu bileşikler, platelet agregasyonunun inhibitörleridir ve bu nedenle, tromboembolik bozuklukların tedavisine veya önlenmesine yönelik ilaçlar olarak kullanılabilir.

IPC Classes
C07D 519/00A61K 31/5025A61P 7/02A61K 31/433C07D 487/04C07D 513/04A61K 31/4355
Parties
Inventor
Jacques Banvılle C/O Université De Montréal 2900 Édouard-Montpetit Boulevard Montréal, Québec H3t 1j4 Kanada Roger Rémıllard 13 Des Cèdres Avenue Napierville, Québec J0j 1l0 Kanada Edward H. Ruedıger C/O Université De Montréal 2900 Édouard-Montpetit Boulevard Montréal, Québec H3t 1j4 Kanada Danıel H. Deon C/O Université De Montréal 2900 Édouard-Montpetit Boulevard Montréal, Québec H3t 1j4 Kanada Marc Gagnon C/O Université De Montréal 2900 Édouard-Montpetit Boulevard Montréal, Québec H3t 1j4 Kanada Laurence Dubé C/O Université De Montréal 2900 Édouard-Montpetit Boulevard Montréal, Québec H3t 1j4 Kanada M. Mıchael Mıller C/O Bristol-Myers Squibb Company Route 206 And Province Line Road Princeton, Nj 08543 A.B.D. Eldon Scott Prıestley C/O Bristol-Myers Squibb Company 311 Pennington- Rocky Hill Road Pennington, New Jersey 08534 A.B.D. Shoshana L. Posy C/O Bristol-Myers Squibb Company Route 206 And Province Line Road Pennington, New Jersey 08543 A.B.D. Brad D. Maxwell C/O Bristol-Myers Squibb Company Route 206 And Province Line Road Pennington, New Jersey 08543 A.B.D. Pancras C. Wong C/O Bristol-Myers Squibb Company 311 Pennington- Rocky Hill Road Pennington, New Jersey 08534 A.B.D. R. Mıchael Lawrence C/O Bristol-Myers Squibb Company 311 Pennington- Rocky Hill Road Pennington, Nj 08534 A.B.D. Julıa Guy C/O Université De Montréal 2900 Édouard-Montpetit Boulevard Montréal, Québec H3t 1j4 Kanada
Rights Holder
Brıstol-Myers Squıbb Company Route 206 And Province Line Road Princeton, Nj 08543 A.B.D. Unıversıté De Montréal 2900 Boulevard Edouard-Montpetit Montreal, Qc H3t 1j4 Kanada
Attorney
Tolga Çaylak (Dış Patent Marka Tescil Ve Danışmanlık Hiz. Ltd. Şti.) İçerenköy Değirmenyolu Cad. No:12/7 K:5 Ataşehir/İstanbul

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