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European Patent (TR Translation)

Muskarinik M1 Reseptör Agonistleri Olarak Bisiklik Aza Bileşikleri.

Invention Abstract

Bu buluş, muskarinik M1 reseptörünün ve/veya M4 reseptörünün agonistleri olan ve muskarinik M1/M4 reseptör aracılı hastalıkların tedavisinde faydalı olan bileşiklere ilişkindir. Ayrıca bileşikleri ve bileşiklerin terapötik kullanımlarını içeren farmasötik bileşimler sağlanmaktadır. Bileşikler formül 1'egöre bileşikleri veya bunların tuzlarını içerir; burada Q R1, R2, R3 ve R4 tanımlandığı gibidir.

IPC Classes
C07D 401/14C07D 471/04C07D 401/04C07D 413/14A61K 31/454C07D 417/14C07D 409/14C07D 405/14C07D 491/107
Parties
Inventor
Gıles Albert Brown C/O Heptares Therapeutics Limited Biopark Broadwater Road Welwyn Garden City Hertfordshire Al7 3ax / İngiltere Julıe Elaıne Cansfıeld C/O Heptares Therapeutics Limited Biopark Broadwater Road Welwyn Garden City Hertfordshire Al7 3ax / İngiltere Mıles Stuart Congreve C/O Heptares Therapeutics Limited Biopark Broadwater Road Welwyn Garden City Hertfordshire Al7 3ax / İngiltere Barry John Teobald C/O Heptares Therapeutics Limited Biopark Broadwater Road Welwyn Garden City Hertfordshire Al7 3ax / İngiltere Mark Pıckworth C/O Heptares Therapeutics Limited Biopark Broadwater Road Welwyn Garden City Hertfordshire Al7 3ax / İngiltere Mark Davıd Rackham C/O Heptares Therapeutics Limited Biopark Broadwater Road Welwyn Garden City Hertfordshire Al7 3ax / İngiltere Benjamın Gerald Tehan C/O Heptares Therapeutics Limited Biopark Broadwater Road Welwyn Garden City Hertfordshire Al7 3ax / İngiltere Mıchael Alıstaır O'brıen C/O Heptares Therapeutics Limited Biopark Broadwater Road Welwyn Garden City Hertfordshire Al7 3ax / İngiltere
Rights Holder
Heptares Therapeutıcs Lımıted Biopark Broadwater Road Welwyn Garden City, Hertfordshire Al7 3ax / İngiltere
Attorney
Hande Mumcuoğlu (Mumcuoğlu Ve Ark Patent Ve Marka Dan. Ltd. Şti.) Mutlukent Mah. Mutluköy Sitesi 1943. Cad. No:10 06800 - Çankaya/Ankara

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